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Regioselective Introduction of Electrophiles into Piperidine Derivatives at the 4-Position


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Title: Regioselective Introduction of Electrophiles into Piperidine Derivatives at the 4-Position
Authors: Onomura, Osamu / Fujimura, Noriyuki / Oda, Takahisa / Matsumura, Yoshihiro / Demizu, Yosuke
Issue Date: Sep-2008
Publisher: Japan Institute of Heterocyclic Chemistry
Citation: Heterocycles, 76(1), pp.177-182; 2008
Abstract: Regioselective introduction of various electrophiles (aldehydes, ketones, and imines) into piperidine skeleton at the 4-position was achieved with a catalytic amount of Pd(OAc)2/PPh3 in the presence of excess Et2Zn. In addition, enantioselective introduction of benzaldehyde into piperidine derivatives was accomplished by using chiral phosphine ligand with moderate enantioselectivity.
URI: http://hdl.handle.net/10069/21989
ISSN: 03855414
DOI: 10.3987/COM-08-S(N)26
Rights: Copyright © 2008 The Japan Institute of Heterocyclic Chemistry
Type: Journal Article
Text Version: author
Appears in Collections:Articles in academic journal

Citable URI : http://hdl.handle.net/10069/21989

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